| S/N | Cas | Name | For APIs |
| 1 | 551-93-9 | 2-Aminoacetophenone | Linagliptin |
| 2 | 109113-72-6 | 2-(Chloromethyl)-4-methylquinazoline | Linagliptin |
| 3 | 1350653-26-7 | 5-fluoro-1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridine-3-carbonitrile | Vericiguat |
| 4 | 1198-97-6 | 4-Phenyl-2-pyrrolidinone | Phenylpiracetam |
| 5 | 52450-32-5 | Ethyl 2-oxo-4-phenylpyrrolidine-3-carboxylate | Phenylpiracetam |
| 6 | 77519-55-2 | 2-oxo-4-phenyl-3-pyrrolidinecarboxylicacid | Phenylpiracetam |
| 7 | 402-43-7 | 4-Bromobenzotrifluoride | / |
| 8 | 871239-18-8 | 2-Amino-5-cyano-3-methylbenzoic acid | cyantraniliprole |
| 9 | 90319-52-1 | (R)-(-)-4-Phenyl-2-oxazolidinone | Ezetimibe |
| 10 | 850012-44-1 | 4-bromo-2-tert-butylphenylamine | / |
| 11 | 1062580-52-2 | (3R,4R)-1-benzyl-N,4-dimethylpiperidin-3-amine dihydrochloride | Tofacitinib |
| 12 | 3680-69-1 | 4-Chloro-7H-pyrrolo[2,3-d]pyrimidine | Tofacitinib |
| 13 | 1187595-85-2 | 2-(1-(ethylsulfonyl)azetidin-3-ylidene)acetonitrile | Baricitinib |
| 14 | 269410-08-4 | 4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole | Baricitinib |
| 15 | 1792190-72-7 | tert-butyl (2S,5R)-5-amino-2-methylpiperidine-1- carboxylate | Ritlecitinib |
| 16 | 80875-98-5 | (2S,3aS,7aS)-Octahydro-1H-indole-2-carboxylic Acid | prindopril |
| 17 | 82834-12-6 | N-[(S)-1-Carbethoxy-1-butyl]-(S)-alanine | prindopril |
| 18 | 6485-55-8 | Cis-2,6-Dimethylmorpholine | Amorolfine |
| 19 | 1563-56-0 | 2-(2-AMINO-5-BROMOBENZOYL) PYRIDINE | Bromazepam |
| 20 | 881674-56-2 | 5-(2-Fluorophenyl)-1H-pyrrole-3-carbaldehyde | Vonoprazan |
| 21 | 739364-95-5 | 2-Methylpyrazolo[1,5-a]pyriMidine-6-carboxylic acid | Anagliptin |
| 22 | 39713-40-1 | 7,8-dihydro-5H-cyclohepta[b]pyridine-5,9(6H)-dione | Rimegepant |
| 23 | 38573-88-5 | 2,3-Difluorobromobenzene | Rimegepant |
| 24 | 7531-52-4 | L-Prolinamide | Vildagliptin |
| 25 | 207557-35-5 | (2S)-1-(Chloroacetyl)-2-pyrrolidinecarbonitrile | Vildagliptin |
| 26 | 13081-18-0 | Ethyl trifluoropyruvate | / |
| 27 | 51067-38-0 | 4-Phenoxyphenyl boronic acid | Ibrutinib |
| 28 | 25487-66-5 | 3-Carboxyphenyl boronic acid | Eltrombopag |
| 29 | 220210-56-0 | 3-(Tert-butoxycarbonyl)phenyl boronic acid | Lumacaftor |
| 30 | 1131-52-8 | 3-Ethoxy-4-methoxybenzaldehyde | Apremilast |
| 31 | 60758-86-3 | 3-Ethoxy-4-methoxybenzonitrile | Apremilast |
| 32 | 51-21-8 | 5-Fluorouracil | Tegafur |
| 33 | 106-40-1 | 4-Bromoaniline | Bedaquiline |
| 34 | 316146-27-7 | N-(4-bromophenyl)-3-phenylpropanamide | Bedaquiline |
| 35 | 2713-34-0 | 3,5-Difluorophenol | Tegoprazan |
| 36 | 87-63-8 | 2-Chloro-6-methylaniline | Bosutinib |
| 37 | 5332-25-2 | 6-Bromoquinoline | Capmatinib |
| 38 | 761446-44-0 | 1-Methylpyrazole-4-boronic acid pinacol ester | New Drug |
| 39 | 415965-24-1 | 4-Bromo-2-fluoro-5-methylbenzoicacid | New Drug |
| 40 | 558-13-4 | Carbon bromide | New Drug |
| 41 | 667-27-6 | ethylbrom(difluor)acetat | Gemcitabine |
| 42 | 15513-48-1 | 4-Chloro-2,6-dimethyl-3-nitropyridine | Grapiprant |
| 43 | 94838-59-2 | [2-(4-Amino-phenyl)-ethyl]-carbamic acid tert-butyl ester | Grapiprant |
| 44 | 35480-52-5 | 2,5-Bis(2,2,2-trifluoroethoxy)benzoic Acid | Flecainide |